Methylphenidate Extended Release (Concerta)

Stimulantprescriptionoral · inferred

Osmotic-release methylphenidate tablet with an initial overcoat dose followed by controlled ascending delivery. The tablet must be swallowed whole.

Projected serum levels — 36 mg, once daily

Methylphenidate Extended Release (Concerta)
Methylphenidate Extended Release (Concerta) modeled serum levels, 36 mg once daily over 15 days Population-based pharmacokinetic estimate. Steady state reached after approximately 1 days. 0 1.3 2.5 3.8 5 Day 0 Day 4 Day 8 Day 11 Day 15 Time on a regular schedule ≈ steady state · day 1

Maintenance schedule: 36 mg once daily (oral).

Modeled steady state after ~1 days: peak ≈ 4.6 mg, trough ≈ 0.37 mg body load. Population-based estimate over 15 days for a 36 mg dose at a 70 kg reference body mass — the interactive app scales curves to your doses, timing, and body mass.

Key facts

Category
Stimulant
Route modeled
Oral
Model confidence
inferred
Half-life
3.6 h
Common dose
36 mg
Suggested maximum
72 mg/day
Reference dose range
18–72 mg (single dose)
Suggested cadence
once daily
Validated against
36 mg oral — Cmax 0.009 mg/L at 6.5 h

Research behind this entry

  1. Methylphenidate for children and adolescents with attention deficit hyperactivity disorder (ADHD) Storebø OJ et al. · Cochrane Database of Systematic Reviews, 2015 DOI

    Cochrane review of 185 RCTs found methylphenidate improves teacher-rated ADHD symptoms and general behavior in children, though evidence quality was low due to risk of bias.

  2. Comparative efficacy and tolerability of medications for attention-deficit hyperactivity disorder in children, adolescents, and adults: a systematic review and network meta-analysis Cortese S et al. · Lancet Psychiatry, 2018 DOI

    Landmark network meta-analysis of 133 RCTs found methylphenidate was the preferred first-choice pharmacotherapy for ADHD in children/adolescents (best efficacy-tolerability balance); amphetamines preferred in adults.

2 published studies referenced in the app, each with a plain-language summary.