Hypericin

Naphthodianthrone

Hypericin is a photoreactive constituent of St. John's wort. Pure hypericin and standardized botanical extracts have different co-constituents and kinetics.

Pharmacokinetic model

A route-level PK model for hypericin is being prepared from published data. Dosing references, studies, and documented interactions are below; the app catalog is updated as models are validated.

Key facts

Category
Naphthodianthrone
Suggested cadence
once daily

Research behind this entry

  1. Pharmacokinetics, safety, and antiviral effects of hypericin, a derivative of St. John's wort plant, in patients with chronic hepatitis C virus infection Jacobson JM, Feinman L, Liebes L, Ostrow N, Koslowski V, Tobia A, Cabana BE, Lee D, Spritzler J, Prince AM · Antimicrobial Agents and Chemotherapy, 2001 DOI

    Nineteen patients received 0.05 or 0.10 mg/kg/day pure hypericin for eight weeks. No meaningful antiviral effect occurred, and phototoxic reactions affected most participants at the higher dose.

1 published study referenced in the app, each with a plain-language summary.